Flumazenil Basic information
Product Name: Flumazenil
Synonyms: ethyl 8-fluoro-5-methyl-6-oxo-5,6-dihydro-4h-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate;FLUMAZENIL;8-FLUORO-5,6-DIHYDRO-5-METHYL-6-OXO-4H-IMIDAZO[1,5-A][1,4]BENZO-DIAZEPINE-3-CARBOXYLIC ACID ETHYL ESTER;8-FLUORO-5,6-DIHYDRO-5-METHYL-6-OXO-4H-IMIDAZO[1,5-A][1,4]BENZODIAZEPINE-3-CARBOXYLIC ACID ETHYL EST;4H-IMIDAZO[1,5-A][1,4]BENZODIAZEPINE-3-CARBOXYLIC ACID, 8-FLUORO-5,6-DIHYDRO-5-METHYL-6-OXO-, ETHYL ESTER;RO 15-1788;Flumazenil、Flumazepil;FlumazenilUsDmf
CAS: 78755-81-4
MF: C15H14FN3O3
MW: 303.29
Flumazenil Chemical Properties
mp 201-203°C
storage temp. 2-8°C
form solid
color white
Water Solubility 128 mg/L
CAS DataBase Reference 78755-81-4(CAS DataBase Reference)
NIST Chemistry Reference Flumazenil(78755-81-4)
Flumazenil Usage And Synthesis
Chemical Properties Colourless crystals
Usage Imidazodiazepine which selectively blocks the central effects of classic benzodiazepines. It is used as benzodiazepine antagonist.
Usage beta-blocker, antihypertensive
Usage benzodiazepine antagonist sedation reversal drug
Biological Activity Benzodiazepine antagonist, non-selective for α 1, α 2, α 3 or α 5-containing GABA A receptors. Centrally active upon systemic administration in vivo .